6-Methylenedihydrodesoxymorphine
A semi-synthetic opioid analgesic
| 6-Methylenedihydrodesoxymorphine | |
|---|---|
| |
| INN | |
| Drug class | |
| Routes of administration | |
| Pregnancy category | |
| Bioavailability | |
| Metabolism | |
| Elimination half-life | |
| Excretion | |
| Legal status | |
| CAS Number | 2033-56-3 |
| PubChem | 5462500 |
| DrugBank | |
| ChemSpider | 4576590 |
| KEGG | |
6-Methylenedihydrodesoxymorphine is a semi-synthetic opioid analgesic derived from morphine. It is a potent analgesic with effects similar to other opioids, acting primarily on the central nervous system to relieve pain.
Chemical Structure[edit | edit source]
6-Methylenedihydrodesoxymorphine is a derivative of morphine, with a methylene group replacing the 6-hydroxy group. This modification results in a compound with increased potency compared to morphine. The chemical structure is characterized by the presence of a morphinan backbone, which is common to many opioid compounds.
Pharmacology[edit | edit source]
6-Methylenedihydrodesoxymorphine acts as an agonist at the mu-opioid receptor, which is responsible for its analgesic effects. The binding of the compound to these receptors inhibits the transmission of pain signals in the nervous system. Like other opioids, it can produce side effects such as respiratory depression, constipation, and euphoria.
Synthesis[edit | edit source]
The synthesis of 6-Methylenedihydrodesoxymorphine involves the chemical modification of morphine. The process typically includes the introduction of a methylene group at the 6-position of the morphine molecule. This synthetic pathway is part of the broader field of opioid chemistry, which explores the creation of new opioid derivatives with varying properties.
Medical Use[edit | edit source]
While 6-Methylenedihydrodesoxymorphine is not commonly used in clinical practice, its study provides valuable insights into the development of new analgesics. Research into such compounds aims to find opioids with improved safety profiles and reduced potential for addiction.
Legal Status[edit | edit source]
As with many opioids, 6-Methylenedihydrodesoxymorphine is subject to strict regulatory control due to its potential for abuse and addiction. It is classified under various national and international drug control laws.
Related pages[edit | edit source]
Gallery[edit | edit source]
Chemical structure of 6-Methylenedihydrodesoxymorphine
6-Methylenedihydrodesoxymorphine[edit | edit source]
6-Methylenedihydrodesoxymorphine structure
Search WikiMD
Ad.Tired of being Overweight? Try W8MD's physician weight loss program.
Semaglutide (Ozempic / Wegovy and Tirzepatide (Mounjaro / Zepbound) available.
Advertise on WikiMD
|
WikiMD's Wellness Encyclopedia |
| Let Food Be Thy Medicine Medicine Thy Food - Hippocrates |
Translate this page: - East Asian
中文,
日本,
한국어,
South Asian
हिन्दी,
தமிழ்,
తెలుగు,
Urdu,
ಕನ್ನಡ,
Southeast Asian
Indonesian,
Vietnamese,
Thai,
မြန်မာဘာသာ,
বাংলা
European
español,
Deutsch,
français,
Greek,
português do Brasil,
polski,
română,
русский,
Nederlands,
norsk,
svenska,
suomi,
Italian
Middle Eastern & African
عربى,
Turkish,
Persian,
Hebrew,
Afrikaans,
isiZulu,
Kiswahili,
Other
Bulgarian,
Hungarian,
Czech,
Swedish,
മലയാളം,
मराठी,
ਪੰਜਾਬੀ,
ગુજરાતી,
Portuguese,
Ukrainian
Medical Disclaimer: WikiMD is not a substitute for professional medical advice. The information on WikiMD is provided as an information resource only, may be incorrect, outdated or misleading, and is not to be used or relied on for any diagnostic or treatment purposes. Please consult your health care provider before making any healthcare decisions or for guidance about a specific medical condition. WikiMD expressly disclaims responsibility, and shall have no liability, for any damages, loss, injury, or liability whatsoever suffered as a result of your reliance on the information contained in this site. By visiting this site you agree to the foregoing terms and conditions, which may from time to time be changed or supplemented by WikiMD. If you do not agree to the foregoing terms and conditions, you should not enter or use this site. See full disclaimer.
Credits:Most images are courtesy of Wikimedia commons, and templates, categories Wikipedia, licensed under CC BY SA or similar.
Contributors: Prab R. Tumpati, MD
