Cyprenorphine

Cyprenorphine is an opioid analgesic that was developed in the 1960s. It is a potent antagonist of the mu-opioid receptor, and has been used in scientific research to help understand the function of this receptor.

History

Cyprenorphine was first synthesized in the 1960s by the pharmaceutical company Hoffmann-La Roche. It was developed as part of a series of related drugs that also includes buprenorphine and diprenorphine, which are still in use today.

Pharmacology

Cyprenorphine acts as an antagonist at the mu-opioid receptor, which is the primary target of most opioid analgesics. It has a high affinity for this receptor, and can effectively block the effects of other opioids. This has made it a useful tool in scientific research, as it can be used to study the effects of opioids on the body and to develop new treatments for opioid addiction.

Medical uses

While cyprenorphine is not commonly used in clinical practice, it has been used in scientific research to study the function of the mu-opioid receptor. It has also been used to develop new treatments for opioid addiction, as it can effectively block the effects of other opioids.

Side effects

Like all opioids, cyprenorphine can cause a range of side effects. These can include nausea, vomiting, constipation, and respiratory depression. It can also cause physical dependence and withdrawal symptoms if used for a long period of time.

See also

• Opioid
• Mu-opioid receptor
• Buprenorphine
• Diprenorphine

Cyprenorphine Resources
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