Mepiprazole

From WikiMD.com Medical Encyclopedia

Anxiolytic drug


Mepiprazole
INN
Drug class
Routes of administration
Pregnancy category
Bioavailability
Metabolism
Elimination half-life
Excretion
Legal status
CAS Number
PubChem
DrugBank
ChemSpider
KEGG


Mepiprazole is a pharmacological compound that was developed as an anxiolytic drug. It belongs to the class of imidazole derivatives and has been studied for its potential effects on anxiety and related disorders.

Chemical Structure[edit | edit source]

Chemical structure of Mepiprazole

Mepiprazole is chemically known as 4-methyl-2-(phenylmethyl)-1H-imidazole. The structure consists of an imidazole ring, which is a five-membered ring containing two nitrogen atoms, with a methyl group and a phenylmethyl group attached. This structure is significant as it influences the drug's pharmacological properties and its interaction with biological targets.

Pharmacology[edit | edit source]

Mepiprazole acts primarily as an anxiolytic, meaning it is used to reduce anxiety. The exact mechanism of action is not fully understood, but it is believed to involve modulation of neurotransmitter systems in the brain, particularly those involving serotonin and dopamine. These neurotransmitters play a crucial role in mood regulation and anxiety.

Clinical Use[edit | edit source]

Mepiprazole was investigated for its potential use in treating anxiety disorders. However, it is not widely used in clinical practice today. The development of newer anxiolytic drugs with more favorable safety profiles and efficacy has overshadowed its use.

Side Effects[edit | edit source]

As with many anxiolytic drugs, mepiprazole may cause side effects. Common side effects include drowsiness, dizziness, and nausea. In some cases, more severe side effects such as allergic reactions or cardiovascular issues may occur.

Research and Development[edit | edit source]

Research into mepiprazole has provided insights into the development of anxiolytic drugs and the role of imidazole derivatives in pharmacology. Although it is not a major drug in current therapeutic use, it has contributed to the understanding of anxiety treatment.

Related Pages[edit | edit source]

WikiMD
Navigation: Wellness - Encyclopedia - Health topics - Disease Index‏‎ - Drugs - World Directory - Gray's Anatomy - Keto diet - Recipes

Search WikiMD

Ad.Tired of being Overweight? Try W8MD's physician weight loss program.
Semaglutide (Ozempic / Wegovy and Tirzepatide (Mounjaro / Zepbound) available.
Advertise on WikiMD

WikiMD's Wellness Encyclopedia

Let Food Be Thy Medicine
Medicine Thy Food - Hippocrates

Medical Disclaimer: WikiMD is not a substitute for professional medical advice. The information on WikiMD is provided as an information resource only, may be incorrect, outdated or misleading, and is not to be used or relied on for any diagnostic or treatment purposes. Please consult your health care provider before making any healthcare decisions or for guidance about a specific medical condition. WikiMD expressly disclaims responsibility, and shall have no liability, for any damages, loss, injury, or liability whatsoever suffered as a result of your reliance on the information contained in this site. By visiting this site you agree to the foregoing terms and conditions, which may from time to time be changed or supplemented by WikiMD. If you do not agree to the foregoing terms and conditions, you should not enter or use this site. See full disclaimer.
Credits:Most images are courtesy of Wikimedia commons, and templates, categories Wikipedia, licensed under CC BY SA or similar.

Contributors: Prab R. Tumpati, MD