Protonitazepyne
A synthetic opioid analgesic
| Protonitazepyne | |
|---|---|
| |
| INN | |
| Drug class | |
| Routes of administration | |
| Pregnancy category | |
| Bioavailability | |
| Metabolism | |
| Elimination half-life | |
| Excretion | |
| Legal status | |
| CAS Number | |
| PubChem | |
| DrugBank | |
| ChemSpider | |
| KEGG | |
Protonitazepyne is a synthetic opioid analgesic that belongs to the benzimidazole class of compounds. It is structurally related to other opioids such as etazene and isotonitazene, which are known for their potent analgesic effects. Protonitazepyne has gained attention due to its potential for abuse and its role in the opioid epidemic.
Chemical Structure[edit | edit source]
Protonitazepyne is characterized by its unique chemical structure, which includes a benzimidazole core. The structure is depicted in the image to the right. This core is responsible for its interaction with the mu-opioid receptor, which mediates its analgesic effects.
Pharmacology[edit | edit source]
Protonitazepyne acts primarily as a mu-opioid receptor agonist. This receptor is part of the opioid receptor family, which also includes the delta-opioid receptor and the kappa-opioid receptor. Activation of the mu-opioid receptor leads to analgesia, euphoria, and respiratory depression, which are characteristic effects of opioid compounds.
Medical Use[edit | edit source]
Currently, Protonitazepyne is not approved for medical use. Its potent analgesic properties suggest potential applications in pain management, but concerns about its safety and abuse potential have limited its development.
Side Effects[edit | edit source]
The side effects of Protonitazepyne are similar to those of other opioids and include:
- Respiratory depression
- Constipation
- Nausea
- Sedation
- Euphoria
Legal Status[edit | edit source]
Due to its potential for abuse and lack of approved medical use, Protonitazepyne is classified as a controlled substance in many jurisdictions. It is subject to strict regulations to prevent misuse and illegal distribution.
Related Compounds[edit | edit source]
Protonitazepyne is related to several other synthetic opioids, including:
Related pages[edit | edit source]
Protonitazepyne
Search WikiMD
Ad.Tired of being Overweight? Try W8MD's physician weight loss program.
Semaglutide (Ozempic / Wegovy and Tirzepatide (Mounjaro / Zepbound) available.
Advertise on WikiMD
|
WikiMD's Wellness Encyclopedia |
| Let Food Be Thy Medicine Medicine Thy Food - Hippocrates |
Translate this page: - East Asian
中文,
日本,
한국어,
South Asian
हिन्दी,
தமிழ்,
తెలుగు,
Urdu,
ಕನ್ನಡ,
Southeast Asian
Indonesian,
Vietnamese,
Thai,
မြန်မာဘာသာ,
বাংলা
European
español,
Deutsch,
français,
Greek,
português do Brasil,
polski,
română,
русский,
Nederlands,
norsk,
svenska,
suomi,
Italian
Middle Eastern & African
عربى,
Turkish,
Persian,
Hebrew,
Afrikaans,
isiZulu,
Kiswahili,
Other
Bulgarian,
Hungarian,
Czech,
Swedish,
മലയാളം,
मराठी,
ਪੰਜਾਬੀ,
ગુજરાતી,
Portuguese,
Ukrainian
Medical Disclaimer: WikiMD is not a substitute for professional medical advice. The information on WikiMD is provided as an information resource only, may be incorrect, outdated or misleading, and is not to be used or relied on for any diagnostic or treatment purposes. Please consult your health care provider before making any healthcare decisions or for guidance about a specific medical condition. WikiMD expressly disclaims responsibility, and shall have no liability, for any damages, loss, injury, or liability whatsoever suffered as a result of your reliance on the information contained in this site. By visiting this site you agree to the foregoing terms and conditions, which may from time to time be changed or supplemented by WikiMD. If you do not agree to the foregoing terms and conditions, you should not enter or use this site. See full disclaimer.
Credits:Most images are courtesy of Wikimedia commons, and templates, categories Wikipedia, licensed under CC BY SA or similar.
Contributors: Prab R. Tumpati, MD
