Valerylfentanyl

Valerylfentanyl

Chemical structure of Valerylfentanyl

3D model of Valerylfentanyl

Valerylfentanyl is a synthetic opioid analgesic that is an analog of fentanyl. It is part of a class of drugs known as fentanyl analogs, which are designed to mimic the effects of fentanyl, a potent opioid used in pain management.

Chemical Properties

Valerylfentanyl is chemically similar to fentanyl, with the primary difference being the substitution of a valeryl group for the propionyl group found in fentanyl. This modification results in changes to the drug's potency, duration of action, and pharmacokinetics.

Pharmacology

Valerylfentanyl acts as an agonist at the mu-opioid receptor, similar to other opioids. This action is responsible for its analgesic effects as well as its potential for abuse and addiction. The potency of valerylfentanyl is generally lower than that of fentanyl, but it still poses significant risks of overdose and respiratory depression.

Legal Status

Due to its potential for abuse and lack of medical use, valerylfentanyl is classified as a controlled substance in many jurisdictions. In the United States, it is listed as a Schedule I substance under the Controlled Substances Act, indicating that it is considered to have a high potential for abuse and no accepted medical use.

Health Risks

The use of valerylfentanyl, like other fentanyl analogs, carries significant health risks. These include the potential for overdose, which can lead to respiratory depression, coma, and death. The drug's potency and the variability in its effects make it particularly dangerous when used illicitly.

Related Pages

• Fentanyl
• Opioid
• Synthetic opioid
• Controlled Substances Act

References

• "Fentanyl and its analogs: A review of the pharmacology and toxicology." Journal of Analytical Toxicology, 2018.
• "The dangers of fentanyl analogs: A public health perspective." American Journal of Public Health, 2019.

Valerylfentanyl

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