Valerylfentanyl

Valerylfentanyl is a potent opioid analgesic that is an analog of fentanyl. It is a designer drug and has been sold online as a research chemical. Valerylfentanyl is less potent than fentanyl, but more potent than morphine.

Chemistry

Valerylfentanyl belongs to the class of organic compounds known as anilides. These are organic heterocyclic compounds derived from acids in which the amino group of an amino acid is replaced by an anilide group.

Pharmacology

Like other opioids, valerylfentanyl binds to and activates the mu-opioid receptor in the brain, spinal cord, and other parts of the body. This leads to an increase in pain threshold and a decrease in the perception of pain.

Effects

The effects of valerylfentanyl are similar to those of other opioids and include analgesia, sedation, and respiratory depression. However, due to its potency, the risk of overdose and death is significantly higher than with other opioids.

Legal Status

Valerylfentanyl is a controlled substance in many countries, including the United States, where it is classified as a Schedule I drug under the Controlled Substances Act. This means it has a high potential for abuse and no accepted medical use.

See Also

• Fentanyl
• Opioid
• Anilides
• Mu-opioid receptor