GW-803430

GW-803430 is a chemical compound that is used in the field of pharmacology. It is a potent and selective agonist for the cannabinoid receptor CB2, with a Ki of 1.2 nM at CB2 and 30 nM at the related CB1 receptor.

Chemical Structure

GW-803430 has a complex chemical structure that includes a pyrazole ring, a phenyl group, and a piperidine ring. The compound is typically synthesized in a laboratory setting using a series of chemical reactions.

Pharmacological Action

GW-803430 acts as an agonist at the CB2 receptor, meaning it binds to this receptor and activates it. This can have a variety of effects in the body, depending on the specific location and function of the CB2 receptor. In general, activation of the CB2 receptor is thought to have anti-inflammatory and analgesic effects.

Potential Therapeutic Uses

Due to its selective action at the CB2 receptor, GW-803430 has been investigated for potential therapeutic uses in conditions such as chronic pain, inflammation, and neurodegenerative diseases. However, more research is needed to fully understand the potential benefits and risks of this compound.

See Also

• Cannabinoid receptor
• Agonist
• Pharmacology