Inaperisone

From WikiMD's Wellness Encyclopedia

Inaperisone is a muscle relaxant used in the treatment of various musculoskeletal disorders. It is a drug that is primarily used in Japan and other parts of Asia. Inaperisone works by blocking the nerve impulses or pain sensations that are sent to the brain, providing relief from discomfort and pain associated with musculoskeletal conditions.

Pharmacology[edit | edit source]

Inaperisone is classified as a centrally acting muscle relaxant. It works by inhibiting the transmission of neurotransmitters in the central nervous system, which in turn reduces muscle tension and spasm. The exact mechanism of action of inaperisone is not fully understood, but it is believed to involve the inhibition of calcium influx into nerve cells, which reduces the release of excitatory neurotransmitters.

Clinical Use[edit | edit source]

Inaperisone is used in the treatment of a variety of musculoskeletal disorders, including muscle spasms, back pain, and fibromyalgia. It is also used in the management of neurological disorders such as multiple sclerosis and spinal cord injury, where muscle spasticity is a common symptom.

Side Effects[edit | edit source]

Like all drugs, inaperisone can cause side effects. The most common side effects of inaperisone include drowsiness, dizziness, and nausea. Less common side effects can include headache, dry mouth, and constipation. In rare cases, inaperisone can cause serious side effects such as allergic reactions, liver damage, and blood disorders.

Contraindications[edit | edit source]

Inaperisone is contraindicated in patients with known hypersensitivity to the drug. It should also be used with caution in patients with liver disease, kidney disease, and in those who are pregnant or breastfeeding.

See Also[edit | edit source]


Muscle relaxants

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Contributors: Prab R. Tumpati, MD