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Template:Antiretroviral drug
From WikiMD.com - Food, Medicine & Wellness Encyclopedia
Antiviral drugs
:
antiretroviral drugs
used against
HIV
(primarily
J05
)
Capsid inhibitors
*
Lenacapavir (LEN)
Entry/fusion inhibitors
(
Discovery and development
)
*
gp41
(
Enfuvirtide (ENF, T-20)
)
◊
CCR5
(
Maraviroc (MVC)
Vicriviroc
†
,
Cenicriviroc
†
,
Leronlimab
†
)
CD4
(
Ibalizumab (IBA)
,
Semzuvolimab
§
)
gp120
(
Fostemsavir (FTR)
)
Integrase inhibitors
(Integrase strand transfer inhibitors (INSTI))
*
Bictegravir (BIC)
Cabotegravir (CAB)
Dolutegravir (DTG)
#
Elvitegravir (EVG)
Raltegravir (RAL)
#
BI 224436
†
MK-2048
†
Maturation inhibitors
*
Bevirimat
†
BMS-955176
§
Fipravirimat
§
Protease Inhibitors (PI)
(
Discovery and development
)
1
st
generation
*
Amprenavir (APV)
‡
Fosamprenavir (FPV)
Indinavir (IDV)
◊
Lopinavir (LPV)
Nelfinavir (NFV)
◊
Ritonavir (RTV)
#
Saquinavir (SQV)
◊
2
nd
generation
*
Atazanavir (ATV)
°
#
Darunavir (DRV)
°
#
Tipranavir (TPV)
◊
TMC-310911
§
#
WHO-EM
‡
Withdrawn
from market
Clinical trials
:
†
Phase III
§
Never to phase III
°
DHHS
recommended
initial regimen options
.
◊
Formerly or rarely used agent.
Category
:
Drug templates by ATC