Isotonitazepyne
Overview[edit | edit source]
Isotonitazepyne is a synthetic opioid analgesic that belongs to the benzimidazole class of compounds. It is structurally related to other opioids such as etonitazene and is known for its potent analgesic properties. Isotonitazepyne has been the subject of research due to its potential use in pain management, but it also poses significant risks of abuse and addiction.
Chemical Structure[edit | edit source]
Isotonitazepyne is characterized by its unique chemical structure, which includes a benzimidazole core. The presence of this core is a defining feature of the nitazene class of opioids. The chemical structure of Isotonitazepyne is depicted in the adjacent image, highlighting its complex arrangement of atoms that contribute to its pharmacological activity.
Pharmacology[edit | edit source]
Isotonitazepyne acts primarily as a mu-opioid receptor agonist, which is the primary mechanism through which it exerts its analgesic effects. By binding to these receptors, it mimics the action of endogenous opioids, leading to pain relief. However, this action also underlies its potential for abuse and the development of opioid use disorder.
Clinical Use[edit | edit source]
While Isotonitazepyne has been investigated for its potential in pain management, its clinical use is limited due to the high risk of addiction and overdose. It is not approved for medical use in many countries and is often encountered in the context of illicit drug use.
Risks and Side Effects[edit | edit source]
The use of Isotonitazepyne carries significant risks, including respiratory depression, which can be fatal. Other side effects include nausea, vomiting, constipation, and sedation. The risk of overdose is particularly high, especially when used in combination with other central nervous system depressants such as benzodiazepines or alcohol.
Legal Status[edit | edit source]
Due to its potential for abuse and lack of approved medical use, Isotonitazepyne is classified as a controlled substance in many jurisdictions. It is important for healthcare providers and law enforcement to be aware of its presence in the illicit drug market.
Related Pages[edit | edit source]
Search WikiMD
Ad.Tired of being Overweight? Try W8MD's physician weight loss program.
Semaglutide (Ozempic / Wegovy and Tirzepatide (Mounjaro / Zepbound) available.
Advertise on WikiMD
|
WikiMD's Wellness Encyclopedia |
| Let Food Be Thy Medicine Medicine Thy Food - Hippocrates |
Translate this page: - East Asian
中文,
日本,
한국어,
South Asian
हिन्दी,
தமிழ்,
తెలుగు,
Urdu,
ಕನ್ನಡ,
Southeast Asian
Indonesian,
Vietnamese,
Thai,
မြန်မာဘာသာ,
বাংলা
European
español,
Deutsch,
français,
Greek,
português do Brasil,
polski,
română,
русский,
Nederlands,
norsk,
svenska,
suomi,
Italian
Middle Eastern & African
عربى,
Turkish,
Persian,
Hebrew,
Afrikaans,
isiZulu,
Kiswahili,
Other
Bulgarian,
Hungarian,
Czech,
Swedish,
മലയാളം,
मराठी,
ਪੰਜਾਬੀ,
ગુજરાતી,
Portuguese,
Ukrainian
Medical Disclaimer: WikiMD is not a substitute for professional medical advice. The information on WikiMD is provided as an information resource only, may be incorrect, outdated or misleading, and is not to be used or relied on for any diagnostic or treatment purposes. Please consult your health care provider before making any healthcare decisions or for guidance about a specific medical condition. WikiMD expressly disclaims responsibility, and shall have no liability, for any damages, loss, injury, or liability whatsoever suffered as a result of your reliance on the information contained in this site. By visiting this site you agree to the foregoing terms and conditions, which may from time to time be changed or supplemented by WikiMD. If you do not agree to the foregoing terms and conditions, you should not enter or use this site. See full disclaimer.
Credits:Most images are courtesy of Wikimedia commons, and templates, categories Wikipedia, licensed under CC BY SA or similar.
Contributors: Prab R. Tumpati, MD
