Zenazocine

From WikiMD's Wellness Encyclopedia

Zenazocine is a drug that belongs to the benzomorphan class of opioids. It was developed in the 1970s by the pharmaceutical company Sterling Drug. Zenazocine is an opioid analgesic drug, which means it is used to relieve pain. It is also a kappa opioid receptor agonist, which means it binds to and activates kappa opioid receptors in the brain and spinal cord to produce its pain-relieving effects.

History[edit | edit source]

Zenazocine was first synthesized in the 1970s by the pharmaceutical company Sterling Drug. It was developed as part of a series of opioid analgesics, which also included pentazocine and phenazocine. However, unlike these other drugs, zenazocine was never marketed for medical use.

Pharmacology[edit | edit source]

Zenazocine is a kappa opioid receptor agonist. This means it binds to and activates kappa opioid receptors in the brain and spinal cord. Activation of these receptors produces analgesia, or pain relief. However, kappa opioid receptor agonists can also produce side effects such as dysphoria (a state of unease or dissatisfaction), hallucinations, and diuresis (increased urine production).

Side Effects[edit | edit source]

The side effects of zenazocine are similar to those of other kappa opioid receptor agonists. These can include dysphoria, hallucinations, and diuresis. Other potential side effects include nausea, vomiting, and constipation. As with all opioids, there is also the risk of addiction and overdose.

See Also[edit | edit source]

Zenazocine Resources
Wikipedia
WikiMD
Navigation: Wellness - Encyclopedia - Health topics - Disease Index‏‎ - Drugs - World Directory - Gray's Anatomy - Keto diet - Recipes

Search WikiMD

Ad.Tired of being Overweight? Try W8MD's physician weight loss program.
Semaglutide (Ozempic / Wegovy and Tirzepatide (Mounjaro / Zepbound) available.
Advertise on WikiMD

WikiMD's Wellness Encyclopedia

Let Food Be Thy Medicine
Medicine Thy Food - Hippocrates

Medical Disclaimer: WikiMD is not a substitute for professional medical advice. The information on WikiMD is provided as an information resource only, may be incorrect, outdated or misleading, and is not to be used or relied on for any diagnostic or treatment purposes. Please consult your health care provider before making any healthcare decisions or for guidance about a specific medical condition. WikiMD expressly disclaims responsibility, and shall have no liability, for any damages, loss, injury, or liability whatsoever suffered as a result of your reliance on the information contained in this site. By visiting this site you agree to the foregoing terms and conditions, which may from time to time be changed or supplemented by WikiMD. If you do not agree to the foregoing terms and conditions, you should not enter or use this site. See full disclaimer.
Credits:Most images are courtesy of Wikimedia commons, and templates Wikipedia, licensed under CC BY SA or similar.

Contributors: Prab R. Tumpati, MD