2-Hydroxysaclofen
2-Hydroxysaclofen is a pharmacological compound that acts as a selective antagonist for the GABAB receptor. It is structurally related to baclofen, which is a potent GABAB agonist.
Pharmacology[edit | edit source]
2-Hydroxysaclofen is a selective GABAB receptor antagonist, meaning it prevents the action of the neurotransmitter GABA at the GABAB receptor subtype. This is in contrast to the related compound baclofen, which is a potent GABAB agonist.
Chemistry[edit | edit source]
2-Hydroxysaclofen is structurally related to baclofen, with the addition of a hydroxyl group at the 2 position of the molecule.
Research[edit | edit source]
Research into 2-Hydroxysaclofen has been conducted to understand its potential therapeutic uses, particularly in the treatment of GABA-related disorders. However, as of now, it is primarily used in scientific research and is not approved for clinical use.
See also[edit | edit source]
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