SB-242084

SB-242084 is a drug that is used in scientific research. It acts as a selective, non-peptide antagonist at the serotonin 5-HT_2C receptor and has been used in the study of this receptor subtype, given its involvement in a variety of physiological processes.

Pharmacology

SB-242084 has been shown to have a high affinity for the 5-HT_2C receptor, with a pKi of 9.0, and 100–200 fold selectivity over other 5-HT₂ subtypes. It has no appreciable affinity for a wide range of other receptors.

Uses

SB-242084 has been used in a variety of studies investigating the role of the 5-HT_2C receptor in various processes and conditions, including anxiety, depression, schizophrenia, and drug addiction. It has also been used to investigate the receptor's role in feeding behavior and energy homeostasis.

Side Effects

As with any drug, SB-242084 may have side effects. However, as it is primarily used in research rather than in clinical practice, these side effects are not well-documented.

See Also

• 5-HT2C receptor
• Serotonin
• 5-HT2A receptor
• 5-HT2B receptor

References

SB-242084 Resources
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