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Serotonin receptor antagonists
...these antagonists can modulate the mood, anxiety, and other functions that serotonin influences. ==Types of Serotonin Receptors==

3 KB (404 words) - 03:38, 2 April 2024
5-HT3 antagonists
...od, anxiety, and emesis (vomiting). By blocking the 5-HT3 receptors, these antagonists can effectively control nausea and vomiting, making them particularly usefu ...The 5-HT3 receptor is a ligand-gated ion channel, which, when activated by serotonin, allows the flow of positively charged ions into the cell, leading to depol

3 KB (404 words) - 15:45, 23 March 2024
5-HT3
...in]], a neurotransmitter that affects mood, appetite, and sleep. The 5-HT3 receptor is a member of the superfamily of [[ligand-gated ion channels]], which are ...cting pore, which is permeable to sodium, potassium, and calcium ions. The receptor is located on the cell membrane of nerve cells, and is particularly prevale

2 KB (275 words) - 20:54, 25 February 2024
Lubazodone
...|alpha-1]] and [[alpha-2 adrenergic receptor|alpha-2 adrenergic]] and [[H1 receptor|H1 histamine]] receptors. ...|alpha-1]] and [[alpha-2 adrenergic receptor|alpha-2 adrenergic]] and [[H1 receptor|H1 histamine]] receptors.

1 KB (168 words) - 22:12, 25 February 2024
5-HT3 receptor
...rotonin]], a neurotransmitter that affects mood, appetite, and sleep. This receptor is found in the [[central nervous system]] and the [[gastrointestinal tract ...nin receptors, is not a [[G protein-coupled receptor]]. It is a pentameric receptor, meaning it is composed of five subunits. These subunits are arranged symme

2 KB (305 words) - 06:26, 20 February 2024
Discovery and development of serotonin receptor antagonists
'''Discovery and Development of Serotonin Receptor Antagonists''' ...f serotonin at its receptors, which can be therapeutic in conditions where serotonin's effects are undesirable.

3 KB (462 words) - 15:42, 23 March 2024
Lurosetron
...he action of serotonin at the 5-HT3 receptor, a subtype of the [[serotonin receptor]]. ...nervous system. The 5-HT3 receptor is activated by the neurotransmitter [[serotonin]], and its activation is associated with a variety of physiological respons

2 KB (250 words) - 04:43, 6 March 2024
Tropisetron
'''Tropisetron''' is a [[serotonin 5-HT3 receptor antagonist]] used mainly as an [[antiemetic]] to treat [[nausea]] and [[vom ...setron acts as both a selective 5-HT3 receptor antagonist and α7-nicotinic receptor agonist. Tropisetron is a well-tolerated drug with few side effects. Headac

1 KB (149 words) - 18:35, 25 February 2024
Zacopride
...c research. It is classified as a [[5-HT4 receptor]] agonist and a [[5-HT3 receptor]] antagonist. Zacopride has been found to have potent [[antiemetic]] and [[ ...f food through the stomach and intestines. At the same time, it blocks the 5-HT3 receptors, which can help to reduce feelings of nausea and vomiting.

1 KB (163 words) - 22:51, 25 February 2024
Bemesetron
...serotonin, a natural substance that may cause nausea and vomiting, at the 5-HT3 receptors in the brain and gut, thereby preventing these symptoms. ...acological action of bemesetron is primarily through its antagonism of the 5-HT3 receptors. These receptors are involved in the vomiting reflex, and their b

3 KB (399 words) - 20:31, 23 April 2024
Lerisetron
...>'''Lerisetron''' is a [[pharmacological]] agent that is classified as a [[5-HT3 antagonist]]. It is primarily used in the prevention and treatment of [[che ...vomiting. It is a potent and selective [[5-HT3 receptor]] antagonist. The 5-HT3 receptors are located on the nerve terminals of the [[vagus nerve]] in the

2 KB (215 words) - 03:43, 6 March 2024
S-268019
...is a [[pharmacological]] agent that is classified as a [[serotonin]] 5-HT3 receptor antagonist. It is primarily used in the treatment of [[chemotherapy]]-induc ...ctive 5-HT3 receptor antagonist with strong binding affinity for the 5-HT3 receptor.

1 KB (182 words) - 19:10, 8 March 2024
Ricasetron
...ea]] and [[vomiting]] (CINV). Ricasetron works by blocking the action of [[serotonin]], a natural substance in the brain that can cause vomiting. ...se receptors, Ricasetron prevents the activation of the vomiting reflex by serotonin, which is released in large amounts during chemotherapy.

2 KB (216 words) - 04:22, 6 March 2024
Azasetron
'''Azasetron''' is a [[serotonin 5-HT3 receptor antagonist]] used in the prevention and treatment of [[postoperative nausea ...ong and long-lasting antiemetic effect. It works by blocking the action of serotonin, a natural substance in the brain that causes nausea and vomiting.

1 KB (145 words) - 21:46, 25 February 2024
Indisetron
...vative of [[indazole]] and is structurally similar to other 5-HT3 receptor antagonists such as [[ondansetron]] and [[granisetron]]. ...entral nervous system]] and [[gastrointestinal tract]], thereby preventing serotonin from activating these receptors.

2 KB (210 words) - 00:15, 11 March 2024
SR-57227
...bowel syndrome]]. SR-57227 is also used in research to explore the role of 5-HT3 receptors in the brain. ...ct]] and the [[central nervous system]]. The drug inhibits the action of [[serotonin]] at these receptors, which can help to reduce nausea and vomiting, and may

2 KB (247 words) - 22:43, 25 February 2024
5-HT3 agonists
...(PNS). These agents are primarily known for their role in stimulating the 5-HT3 receptors, which can influence various physiological and pathological proce ...ansmitters and have various effects depending on the location of the 5-HT3 receptor within the body.

3 KB (430 words) - 03:35, 2 April 2024
Ramosetron
'''Ramosetron''' is a [[serotonin]] 5-HT3 receptor antagonist used in the treatment and prevention of [[nausea]] and [[vomitin ...elective 5-HT3 receptor antagonist with a strong binding affinity for this receptor.

2 KB (206 words) - 23:10, 25 February 2024
Dazopride
...rders. It is a [[5-HT3 antagonist]], which means it blocks the action of [[serotonin]] in the brain. This can help to reduce feelings of [[nausea]] and [[vomiti ...nding to and blocking the [[5-HT3 receptor]], a specific type of serotonin receptor. This can help to reduce the symptoms of gastrointestinal disorders.

1 KB (201 words) - 23:00, 25 February 2024
5-HT3 antagonist
5-HT3 Antagonists (Setrons) ...signed to inhibit the action of the 5-HT3 receptor, a subtype of serotonin receptor primarily found in the terminals of the vagus nerve and in specific brain r

3 KB (461 words) - 01:38, 15 June 2023