Phenazolam
Phenazolam is a benzodiazepine derivative which was never marketed. It has sedative and anxiolytic effects similar to those produced by other benzodiazepine derivatives, and is around the same potency as chlordiazepoxide.
Pharmacology[edit | edit source]
Phenazolam acts as a GABA agonist to exert its pharmacological effects. Like other benzodiazepines, it enhances the effect of GABA at the GABAA receptor, resulting in sedative, sleep-inducing, anxiolytic, anticonvulsant, and muscle relaxant properties.
Medical Uses[edit | edit source]
Phenazolam has never been marketed for medical use, but it has been sold as a designer drug. It is used recreationally for its sedative and anxiolytic effects.
Side Effects[edit | edit source]
The side effects of Phenazolam are similar to those of other benzodiazepines, and can include drowsiness, dizziness, confusion, and memory impairment. Long-term use can lead to tolerance, dependence, and withdrawal symptoms on discontinuation.
See Also[edit | edit source]
References[edit | edit source]
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