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Template:Targeted cancer therapeutic agents
From WikiMD.com Medical Encyclopedia
v
t
e
Targeted cancer therapy
/
antineoplastic agents
(
L01
)
CI
monoclonal antibodies
("-mab")
Receptor tyrosine kinase
ErbB
:
HER1/EGFR
(
Cetuximab
Panitumumab
)
HER2/neu
(
Pertuzumab
,
Trastuzumab
(
+hyaluronidase
)
Trastuzumab emtansine
Trastuzumab deruxtecan
)
Others for solid tumors
EpCAM
(
Catumaxomab
Edrecolomab
)
VEGF-A
(
Bevacizumab
)
Leukemia
/
lymphoma
lymphoid
:
CD3
(
Glofitamab
,
Elranatamab
,
Mosunetuzumab
),
CD20
(
Glofitamab
Ibritumomab
Mosunetuzumab
Obinutuzumab
Ofatumumab
Rituximab
Tositumomab
),
CD30
(
Brentuximab
),
CD52
(
Alemtuzumab
)
myeloid
:
CD33
(
Gemtuzumab ozogamicin
)
Other
Amivantamab
Atezolizumab
Avelumab
Belantamab mafodotin
Bermekimab
Blinatumomab
Cemiplimab
Daratumumab
Dinutuximab beta
Dostarlimab
Durvalumab
Elotuzumab
Enfortumab vedotin
Inotuzumab ozogamicin
Ipilimumab
Isatuximab
Mirvetuximab soravtansine
Mogamulizumab
Moxetumomab pasudotox
Necitumumab
Nivolumab
Olaratumab
Pembrolizumab
Polatuzumab vedotin
Ramucirumab
Retifanlimab
Tafasitamab
Tyrosine kinase inhibitors
("-nib")
Receptor tyrosine kinase
ErbB
:
HER1/EGFR
(
Afatinib
Brigatinib
Dacomitinib
Erlotinib
Gefitinib
Icotinib
Mobocertinib
Olmutinib
Osimertinib
Rociletinib
Vandetanib
)
HER1/EGFR and
HER2/neu
Lapatinib
Neratinib
Tucatinib
RTK class III
:
C-kit
and
PDGFR
(
Avapritinib
Axitinib
Masitinib
Pazopanib
Ripretinib
Sorafenib
Sunitinib
Toceranib
)
FLT3
(
Lestaurtinib
,
Gilteritinib
(AXL, ALK, LTK))
VEGFR
Axitinib
Cediranib
Fruquintinib
Lenvatinib
Nintedanib
Pazopanib
Regorafenib
Semaxanib
Sorafenib
Sunitinib
Tivozanib
Toceranib
Vandetanib
ALK
Alectinib
Brigatinib
Ceritinib
RET
inhibitors:
Entrectinib
(ALK, ROS1, NTRK),
Futibatinib
(FGFR2),
Infigratinib
,
Larotrectinib
(NTRK),
Pemigatinib
(FGFR),
Pralsetinib
,
Repotrectinib
(ROS1, TRK, ALK),
Selpercatinib
(VEGFR, FGFR),
Vandetanib
(VEGFR, EGFR).
c-MET
inhibitors:
Cabozantinib
(VEGFR),
Capmatinib
,
Crizotinib
(ALK)
Non-receptor
bcr-abl
Asciminib
Bosutinib
Dasatinib
Imatinib
Nilotinib
Ponatinib
Radotinib
Src
(
Bosutinib
Dasatinib
)
Janus kinase
Baricitinib
Fedratinib
Filgotinib
Lestaurtinib
Momelotinib
Pacritinib
Ruxolitinib
MAP2K
Binimetinib
Cobimetinib
Selumetinib
Trametinib
EML4
-
ALK
Crizotinib
Entrectinib
Lorlatinib
Bruton's
Acalabrutinib
Ibrutinib
Pirtobrutinib
Zanubrutinib
Other
fusion protein
against
VEGF
(
Aflibercept
)
proapoptotic
peptide against
ANXA2
and
prohibitin
(
Adipotide
)
exotoxin
against
IL-2
(
Denileukin diftitox
)
mTOR inhibitors
Everolimus
Ridaforolimus
Temsirolimus
hedgehog
inhibitors
Glasdegib
Sonidegib
Vismodegib
CDK inhibitors
Abemaciclib
Dalpiciclib
Palbociclib
Ribociclib
Trilaciclib
KRAS
inhibitors
Adagrasib
Sotorasib
Cabozantinib
Capmatinib
Entrectinib
Erdafitinib
Gilteritinib
Larotrectinib
Lenvatinib
Masitinib
Midostaurin
Nintedanib
Pazopanib
Pemigatinib
Pexidartinib
Quizartinib
Regorafenib
Ripretinib
Sorafenib
Sunitinib
Tebentafusp
Tepotinib
Vandetanib
Venetoclax
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