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Template:Leukotriene signaling modulators
From WikiMD.com - Food, Medicine & Wellness Encyclopedia
Leukotriene
signaling
modulators
Receptor
(
ligands
)
BLT
BLT
1
*
Agonists:
12-HETE
20-Hydroxy-LTB
4
Leukotriene B
4
LY-255283
Antagonists:
20-Carboxy-LTB
4
Amelubant
CGS-23131 (LY-223982)
CGS-25019C
CP-105696
CP-195543
Etalocib
LY-293111
Moxilubant
ONO-4057
RG-14893
RP-69698
SB-209247
SC-53228
Ticolubant
U-75302
ZK-158252
BLT
2
*
Agonists:
12-HETE
12-HHT
12-HpETE
15-HETE
15-HpETE
20-Hydroxy-LTB
4
Leukotriene B
4
Antagonists:
CP-195543
LY-255283
ZK-158252
CysLT
CysLT
1
*
Agonists:
Leukotriene C
4
Leukotriene D
4
Leukotriene E
4
Antagonists:
Ablukast
BAYu9773
BAYu9916
BAYx7195
Cinalukast
FPL-55712
ICI-198615
Iralukast
LY-170680
Masilukast
MK-571
Montelukast
ONO-1078
Pobilukast
Pranlukast
Ritolukast
SKF-104353
SR-2640
Sulukast
Tipelukast
Tomelukast
Verlukast
Zafirlukast
ZD-3523
CysLT
2
*
Agonists:
Leukotriene C
4
Leukotriene D
4
Leukotriene E
4
Antagonists:
BAYu9773
BAYu9916
CysLT
E
*
Agonists:
Leukotriene E
4
Enzyme
(
inhibitors
)
5-LOX
*
2-TEDC
Baicalein
BW-A4C
BW-B70C
Caffeic acid
CDC
CJ-13610
Curcumin
Fenleuton
Hyperforin
Hypericum perforatum
(St. John's Wort)
Meclofenamic acid (meclofenamate)
Minocycline
N-Stearoyldopamine
Timegadine
Zileuton
FLAP
inhibitors:
AM-103
AM-679
BAYx1005
MK-591
MK-886
12-LOX
*
2-TEDC
3-Methoxytropolone
Baicalein
CDC
15-LOX
*
2-TEDC
CDC
Luteolin
PD-146176
LTA
4
H
*
Acebilustat
Captopril
DG-051
Fosinoprilat
JNJ-26993135
SA-6541
SC-57461A
Ubenimex (bestatin)
LTB
4
H
*
17-Octadecynoic acid
Others
*
Precursors:
Linoleic acid
γ-Linolenic acid (gamolenic acid)
Dihomo-γ-linolenic acid
Diacylglycerol
Arachidonic acid
5-HPETE (arachidonic acid 5-hydroperoxide)
Leukotriene A
4
;See also
Receptor/signaling modulators
Prostanoid signaling modulators
Category
:
Drug templates by receptor, channel, or pump