Excitatory amino acid reuptake inhibitor

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An excitatory amino acid reuptake inhibitor (EAARI) is a type of drug which inhibits the reuptake of the excitatory neurotransmitters glutamate and aspartate by blocking one or more of the excitatory amino acid transporters (EAATs)

See also[edit]

Pharmacomodulation

Types

* ♦ Enzyme: Inducer

Inhibitor

♦ Ion channel: Opener
Blocker

♦ Transporter [Reuptake vs Efflux]: Enhancer (RE)
Inhibitor (RI)
Releaser (RA)

♦ Miscellaneous: Precursor
Cofactor

Classes

see Enzyme inhibition

See Ion channel modulators

Receptor &
transporter

Adrenergic	* Adrenergic receptor agonist (α β (1 2)) Adrenergic receptor antagonist (α (1 2) β) Norepinephrine reuptake inhibitor (NRI)
Dopaminergic	* Dopamine receptor agonist Dopamine receptor antagonist Dopamine reuptake inhibitor (DRI)
Histaminergic	* Histamine receptor agonist Histamine receptor antagonist (H₁ H₂ H₃)

* Acetylcholine receptor agonist (Muscarinic

Cannabinoidergic

* Cannabinoid receptor agonist

Cannabinoid receptor antagonist
Endocannabinoid enhancer (eCBE)
Endocannabinoid reuptake inhibitor (eCBRI)

Miscellaneous

* Cofactor (see Enzyme cofactors)

Precursor (see Amino acids)

Glutamate metabolism and transport modulators

* 4-Methylene-L-glutamate

GAH	* BPTES CB-839 DON
AST	* 2-Amino-3-butenoic acid AAOA AMB β-DL -Methylene-aspartate Hydrazinosuccinate
ALT	* β-Chloro-L -alanine L -Cycloserine Propargylglycine
GDH	* AAOA Bithionol Chloroquine EGCG GTP GW5074 Hexachlorophene Hydroxylamine Palmitoyl-CoA Pyridoxal phosphate
GS	* 2-Aminoadipic acid JFD01307SC Methionine sulfoximine Phosphinothricin (glufosinate)

See also: Receptor/signaling modulators • Ionotropic glutamate receptor modulators • Metabotropic glutamate receptor modulators • GABA metabolism and transport modulators

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Excitatory amino acid reuptake inhibitors