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Template:Chemokine receptor modulators
From WikiMD.com - Food, Medicine & Wellness Encyclopedia
Chemokine receptor
modulators
CC
CCR1
*
Agonists:
CCL4 (MIP-1β)
CCL5 (RANTES)
CCL6
CCL9 (CCL10)
CCL14
CCL15
CCL16
CCL23
CCR2
*
Agonists:
CCL2
CCL8
CCL12
CCL16
NAMs:
Cenicriviroc (TAK-652, TBR-652)
CCR3
*
Agonists:
CCL5 (RANTES)
CCL7
CCL11
CCL13
CCL15
CCL18
CCL24
CCL26
CCL28
CCR4
*
Agonists:
CCL3 (MIP-1α)
CCL5 (RANTES)
CCL17
CCL22
Antibodies:
Mogamulizumab
(against CCR4)
CCR5
*
Agonists:
CCL3 (MIP-1α)
CCL4 (MIP-1β)
CCL5 (RANTES)
CCL8
CCL11
CCL13
CCL14
CCL16
NAMs:
Aplaviroc
Cenicriviroc (TAK-652, TBR-652)
INCB009471
Maraviroc
Vicriviroc
Antibodies:
PRO-140
CXC
CXCR1
(IL-8Rα)
*
Agonists:
CXCL6
Emoctakin
Interleukin-8 (CXCL8, GCP-1)
Antagonists:
Navarixin
NAMs:
Ladarixin
Reparixin (repertaxin)
CXCR2
(IL-8Rβ)
*
Agonists:
CXCL1 (MGSA)
CXCL2
CXCL3
CXCL5
CXCL6
CXCL7
Emoctakin
Garnocestim
Interleukin-8 (CXCL8, GCP-1)
Antagonists:
Danirixin
Elubrixin
Navarixin
NAMs:
Ladarixin
Reparixin (repertaxin)
CXCR3
*
Agonists:
CXCL4 (PF4)
CXCL9 (MIG)
CXCL10 (IP-10)
CXCL11 (I-TAC)
Iroplact
Antibodies:
Eldelumab
(against CXCL10)
CXCR4
*
Agonists:
MIF
SDF-1 (CXCL12)
Ubiquitin
Antagonists:
Mavorixafor
Plerixafor (AMD3100)
Antibodies:
Ulocuplumab
(against CXCR4)
CXCR5
*
Agonists:
CXCL13
C (XC)
XCR1
*
Agonists:
Lymphotactin-α (XCL1)
Lymphotactin-β (XCL2)
Antibodies:
Pateclizumab
CX3C
CX3CR1
*
Agonists:
Fractalkine (CX3CL1)
Others
CCBP2
*
Agonists:
CC (β) chemokines
CMKLR1
*
Agonists:
Chemerin
Resolvin E1
Category
:
Drug templates by receptor, channel, or pump