Despropionyl-p-fluorofentanyl

From WikiMD's Wellness Encyclopedia

Despropionyl-p-fluorofentanyl


Despropionyl-p-fluorofentanyl is a synthetic opioid that is an analog of fentanyl. It is also known as 4-Fluorofentanyl and is a potent opioid receptor agonist.

Chemistry[edit | edit source]

Despropionyl-p-fluorofentanyl is a fluorinated analog of fentanyl, a powerful synthetic opioid analgesic that is similar to morphine but is 50 to 100 times more potent. The chemical structure of despropionyl-p-fluorofentanyl is similar to that of fentanyl, but with a fluorine atom added to the phenethyl group.

Pharmacology[edit | edit source]

Despropionyl-p-fluorofentanyl acts as a potent agonist at the mu-opioid receptor. It has a high affinity for this receptor, which is the primary site of action for the most commonly used opioids. The binding of despropionyl-p-fluorofentanyl to the mu-opioid receptor results in a range of effects, including analgesia, sedation, and respiratory depression.

Effects[edit | edit source]

The effects of despropionyl-p-fluorofentanyl are similar to those of other opioids. These include analgesia, sedation, euphoria, and respiratory depression. However, due to its high potency, the risk of overdose and death is significantly higher than with other opioids.

Legal Status[edit | edit source]

Despropionyl-p-fluorofentanyl is a controlled substance in many countries due to its high potential for abuse and addiction. In the United States, it is classified as a Schedule I drug under the Controlled Substances Act.

See Also[edit | edit source]




WikiMD
Navigation: Wellness - Encyclopedia - Health topics - Disease Index‏‎ - Drugs - World Directory - Gray's Anatomy - Keto diet - Recipes

Search WikiMD

Ad.Tired of being Overweight? Try W8MD's physician weight loss program.
Semaglutide (Ozempic / Wegovy and Tirzepatide (Mounjaro / Zepbound) available.
Advertise on WikiMD

WikiMD's Wellness Encyclopedia

Let Food Be Thy Medicine
Medicine Thy Food - Hippocrates

Medical Disclaimer: WikiMD is not a substitute for professional medical advice. The information on WikiMD is provided as an information resource only, may be incorrect, outdated or misleading, and is not to be used or relied on for any diagnostic or treatment purposes. Please consult your health care provider before making any healthcare decisions or for guidance about a specific medical condition. WikiMD expressly disclaims responsibility, and shall have no liability, for any damages, loss, injury, or liability whatsoever suffered as a result of your reliance on the information contained in this site. By visiting this site you agree to the foregoing terms and conditions, which may from time to time be changed or supplemented by WikiMD. If you do not agree to the foregoing terms and conditions, you should not enter or use this site. See full disclaimer.
Credits:Most images are courtesy of Wikimedia commons, and templates Wikipedia, licensed under CC BY SA or similar.

Contributors: Prab R. Tumpati, MD