- Benzathine benzylpenicillin# - Procaine benzylpenicillin# - Phenoxymethylpenicillin (V)# - Propicillin‡ - Pheneticillin‡ - Azidocillin‡ - Clometocillin‡
- Flucloxacillin) - Oxacillin - Nafcillin
- Ampicillin# (Pivampicillin - Hetacillin‡ - Bacampicillin‡ - Lenampicillin - Metampicillin‡ - Talampicillin‡)
- Carbenicillin‡ / Carindacillin‡
- Azlocillin‡
- Antipseudomonal (Doripenem - Imipenem - Meropenem) - Biapenem‡ - Panipenem) - Penems (Faropenem - Ritipenem§
- Cefalexin # - Cefadroxil - Cefapirin - Cefazedone‡ - Cefazaflur‡ - Cefradine‡ - Cefroxadine‡ - Ceftezole‡ - Cefaloglycin‡ - Cefacetrile‡ - Cefalonium‡ - Cefaloridine‡ - Cefalotin
- Cefprozil - Cefuroxime - Cefuroxime axetil - Cefamandole‡ - Cefonicid‡ - Ceforanide‡ - Cefuzonam‡ - Cephamycin (Cefoxitin - Cefotetan - Cefminox‡ - Cefbuperazone‡ - Cefmetazole‡)
- Ceftriaxone# - Cefotaxime# - Antipseudomonal (Ceftazidime# - Cefoperazone) - Cefdinir - Cefcapene - Cefdaloxime - Ceftizoxime - Cefmenoxime - Cefpiramide - Cefpodoxime - Ceftibuten - Cefditoren - Cefotiam‡ - Cefetamet‡ - Cefodizime‡ - Cefpimizole‡ - Cefsulodin‡ - Cefteram‡ - Ceftiolene‡ - Oxacephem (Flomoxef
- Cefozopran‡ - Cefpirome
- Ceftolozane
- Tigemonam‡ - Carumonam‡
- Tazobactam) - Clavam (Clavulanic acid) - non-β-lactam (Avibactam - Durlobactam - Relebactam
- DADAL/AR inhibitors (Cycloserine)
- - lysozyme - Tyrothricin - - Gramicidin - - Tyrocidine - Isoniazid#
DHFR inhibitors - 2,4-Diaminopyrimidine (Brodimoprim - Iclaprim - Ormetoprim - Pyrimethamine - Tetroxoprim - Trimethoprim) Sulfonamides (DHPS inhibitors) Short-acting - Sulfisomidine - Sulfamethizole - Sulfadimidine (Sulfamethazine - Sulfadimerazine - Sulfadimezine) - Sulfapyridine (Sulfasalazine) - Sulfafurazole (Acetyl sulfisoxazole) - Sulfanilamide (Prontosil) - Sulfathiazole (Phthalylsulfathiazole - Succinylsulfathiazole) - Sulfathiourea
Intermediate-acting - Sulfamethoxazole - Sulfadiazine - Sulfamoxole
Long-acting - Sulfadimethoxine - Sulfadoxine - Sulfalene - Sulfametomidine - Sulfametoxydiazine - Sulfamethoxypyridazine - Sulfaperin - Sulfamerazine - Sulfaphenazole - Sulfamazone
Other/ungrouped - Mafenide - Sulfacetamide - Sulfaclozine - Sulfadicramide - Sulfaguanidine - Sulfametrole - Sulfanitran
Combinations - Trimethoprim/sulfamethoxazole - Ormetoprim/sulfadimethoxine - Pyrimethamine/dapsone - Pyrimethamine/sulfadoxine
Other DHPS inhibitors - Acediasulfone - Dapsone - Solasulfone - Sulfoxone
1st Generation - Cinoxacin - Flumequine - Nalidixic acid - Oxolinic acid - Pipemidic acid - Piromidic acid - Rosoxacin
Fluoroquinolones 2nd Gen - Ciprofloxacin - Ofloxacin - Enoxacin - Fleroxacin - Lomefloxacin - Nadifloxacin - Levonadifloxacin - Alalevonadifloxacin - Norfloxacin - Pefloxacin - Rufloxacin
3rd Gen - Levofloxacin - Balofloxacin - Grepafloxacin - Pazufloxacin - Sparfloxacin - Temafloxacin - Tosufloxacin
4th Gen - Besifloxacin - Delafloxacin - Gatifloxacin - Finafloxacin - Gemifloxacin - Moxifloxacin - Clinafloxacin - Garenoxacin - Prulifloxacin - Sitafloxacin - Trovafloxacin - Alatrofloxacin
Veterinary use - Danofloxacin - Difloxacin - Enrofloxacin - Ibafloxacin - Marbofloxacin - Orbifloxacin - Pradofloxacin - Sarafloxacin
Newer non-fluorinated - Nemonoxacin - Ozenoxacin Related (DNA gyrase) - Aminocoumarins (Novobiocin)
Nitroimidazole derivatives - Secnidazole
Rifamycins - Rifampicin - Rifabutin - Rifapentine - Rifaximin - Rifalazil Lipiarmycins - Fidaxomicin